SGC Chemical Probe Citation Timeline




(Last updated on 2026-10-03 - zoom via mouse wheel)
Citation counts from OpenAlex; may be lower than Google Scholar.

Target Class

2OG         
AT         
BRD         
DEHYDR         
E3 ligase         
KDM         
Kinase         
MBT         
PAD         
PMT         
PWWP         
Spindlin         
UBD         
USP         
WD40         
White_Paper         
Yeats         
Target Class Target Probe Date Published Number of Citations
BRD BET family (+)-JQ1 2010-09-01 5038
PMT G9a/GLP UNC638 2011-07-10 540
KDM JMJD3/UTX GSK-J4/J1 2012-08-01 979
PMT PRC2 GSK343 2012-10-09 380
PMT DOT1L SGC0946 2012-12-01 294
MBT L3MBTL3 UNC1215 2013-01-16 174
PMT PRC2 UNC1999 2013-04-08 540
BRD BET PFI-1 2013-04-10 251
2OG PHD2/ELGN-1 IOX2 2013-05-17 117
PMT G9a/GLP UNC0642 2013-11-01 280
PMT G9a/GLP A-366 2014-01-02 190
KDM pan-2-OG IOX1 2014-02-06 80
BRD CBP/p300 SGC-CBP30 2014-06-19 289
PMT SETD7 (R)-PFI-2 2014-09-01 193
PAD PAD4 GSK484 2015-01-26 796
PMT PRMT3 SGC707 2015-02-10 141
BRD BAZ2A,B BAZ2-ICR 2015-02-26 105
PMT SMYD2 LLY-507 2015-03-30 134
BRD BRD9 I-BRD9 2015-04-09 238
BRD BRD7,9 LP99 2015-04-13 125
BRD SMARCA2/4 PFI-3 2015-07-01 282
KDM KDM1A GSK-LSD1 2015-07-13 522
PMT MLL OICR-9429 2015-08-01 295
DEHYDR IDH1 mutant GSK864 2015-10-01 180
BRD CREBBP, EP300 I-CBP112 2015-12-01 233
PMT PRMT5 GSK591 2015-12-01 166
BRD BAZ2A/2B GSK2801 2016-02-01 164
BRD BRD9/7 BI-9564 2016-02-25 228
PMT PRMT type 1 MS023 2016-03-01 308
BRD BRPF1B GSK6853 2016-05-01 67
PMT SMYD2 BAY-598 2016-05-01 91
BRD ATAD2A/B GSK8814 2016-09-01 13
PMT PRMT4/6 MS049 2016-10-01 92
BRD PCAF/GCN5 GSK4027 2017-01-01 105
BRD BRPF1-3 NI-42 2017-01-09 55
BRD PCAF, GCN5 L-Moses 2017-01-16 13
PMT SUV420H1/H2 A-196 2017-03-01 135
PMT PRC2 A-395 2017-04-01 236
BRD BRD1, TAF1 BAY-299 2017-04-12 70
BRD BRPF1-3 NI-57 2017-07-17 40
BRD BRPF1-3 OF-1 2017-08-29 57
BRD BRPF1B PFI-4 2017-08-29 57
AT CREBBP, EP300 A-485 2017-09-01 914
BRD ATAD2A BAY-850 2017-10-18 91
PMT PRMT4 TP-064 2018-04-06 155
PMT PRMT5 LLY-283 2018-04-23 190
Kinase GAK SGC-GAK-1 2018-07-25 72
Yeats MLLT1/3 SGC-iMLLT 2018-10-05 97
BRD pan-BRD Bromosporine 2019-01-21 57
PWWP NSD3 BI-9321 2019-07-08 105
PMT SMYD2 PFI-5 2019-08-15 19
Spindlin SPIN1 VinSpinin 2019-09-24 47
PMT PRMT4 SKI-73 2019-10-28 61
White_Paper Target_2035 Target_2035 2019-11-01 182
PMT PRDM9 MRK-740 2019-12-17 44
PWWP NSD2 UNC6934 2021-02-01 67
PMT PRMT6 SGC6870 2021-02-16 30
PMT SMYD3 BAY-6035 2021-06-21 27
White_Paper CACHE CACHE 2022-02-15 116
USP USP21 BAY-805 2023-02-20 28
UBD HDAC6 SGC-UBD253 2023-07-21 12
Kinase CDKL5 SGC-CAF382-1 2023-07-25 15
Total Citations 16,622