| Target Class | Target | Probe | Date Published | Number of Citations |
|---|---|---|---|---|
| BRD | BET family | (+)-JQ1 | 2010-09-01 | 5038 |
| PMT | G9a/GLP | UNC638 | 2011-07-10 | 540 |
| KDM | JMJD3/UTX | GSK-J4/J1 | 2012-08-01 | 979 |
| PMT | PRC2 | GSK343 | 2012-10-09 | 380 |
| PMT | DOT1L | SGC0946 | 2012-12-01 | 294 |
| MBT | L3MBTL3 | UNC1215 | 2013-01-16 | 174 |
| PMT | PRC2 | UNC1999 | 2013-04-08 | 540 |
| BRD | BET | PFI-1 | 2013-04-10 | 251 |
| 2OG | PHD2/ELGN-1 | IOX2 | 2013-05-17 | 117 |
| PMT | G9a/GLP | UNC0642 | 2013-11-01 | 280 |
| PMT | G9a/GLP | A-366 | 2014-01-02 | 190 |
| KDM | pan-2-OG | IOX1 | 2014-02-06 | 80 |
| BRD | CBP/p300 | SGC-CBP30 | 2014-06-19 | 289 |
| PMT | SETD7 | (R)-PFI-2 | 2014-09-01 | 193 |
| PAD | PAD4 | GSK484 | 2015-01-26 | 796 |
| PMT | PRMT3 | SGC707 | 2015-02-10 | 141 |
| BRD | BAZ2A,B | BAZ2-ICR | 2015-02-26 | 105 |
| PMT | SMYD2 | LLY-507 | 2015-03-30 | 134 |
| BRD | BRD9 | I-BRD9 | 2015-04-09 | 238 |
| BRD | BRD7,9 | LP99 | 2015-04-13 | 125 |
| BRD | SMARCA2/4 | PFI-3 | 2015-07-01 | 282 |
| KDM | KDM1A | GSK-LSD1 | 2015-07-13 | 522 |
| PMT | MLL | OICR-9429 | 2015-08-01 | 295 |
| DEHYDR | IDH1 mutant | GSK864 | 2015-10-01 | 180 |
| BRD | CREBBP, EP300 | I-CBP112 | 2015-12-01 | 233 |
| PMT | PRMT5 | GSK591 | 2015-12-01 | 166 |
| BRD | BAZ2A/2B | GSK2801 | 2016-02-01 | 164 |
| BRD | BRD9/7 | BI-9564 | 2016-02-25 | 228 |
| PMT | PRMT type 1 | MS023 | 2016-03-01 | 308 |
| BRD | BRPF1B | GSK6853 | 2016-05-01 | 67 |
| PMT | SMYD2 | BAY-598 | 2016-05-01 | 91 |
| BRD | ATAD2A/B | GSK8814 | 2016-09-01 | 13 |
| PMT | PRMT4/6 | MS049 | 2016-10-01 | 92 |
| BRD | PCAF/GCN5 | GSK4027 | 2017-01-01 | 105 |
| BRD | BRPF1-3 | NI-42 | 2017-01-09 | 55 |
| BRD | PCAF, GCN5 | L-Moses | 2017-01-16 | 13 |
| PMT | SUV420H1/H2 | A-196 | 2017-03-01 | 135 |
| PMT | PRC2 | A-395 | 2017-04-01 | 236 |
| BRD | BRD1, TAF1 | BAY-299 | 2017-04-12 | 70 |
| BRD | BRPF1-3 | NI-57 | 2017-07-17 | 40 |
| BRD | BRPF1-3 | OF-1 | 2017-08-29 | 57 |
| BRD | BRPF1B | PFI-4 | 2017-08-29 | 57 |
| AT | CREBBP, EP300 | A-485 | 2017-09-01 | 914 |
| BRD | ATAD2A | BAY-850 | 2017-10-18 | 91 |
| PMT | PRMT4 | TP-064 | 2018-04-06 | 155 |
| PMT | PRMT5 | LLY-283 | 2018-04-23 | 190 |
| Kinase | GAK | SGC-GAK-1 | 2018-07-25 | 72 |
| Yeats | MLLT1/3 | SGC-iMLLT | 2018-10-05 | 97 |
| BRD | pan-BRD | Bromosporine | 2019-01-21 | 57 |
| PWWP | NSD3 | BI-9321 | 2019-07-08 | 105 |
| PMT | SMYD2 | PFI-5 | 2019-08-15 | 19 |
| Spindlin | SPIN1 | VinSpinin | 2019-09-24 | 47 |
| PMT | PRMT4 | SKI-73 | 2019-10-28 | 61 |
| White_Paper | Target_2035 | Target_2035 | 2019-11-01 | 182 |
| PMT | PRDM9 | MRK-740 | 2019-12-17 | 44 |
| PWWP | NSD2 | UNC6934 | 2021-02-01 | 67 |
| PMT | PRMT6 | SGC6870 | 2021-02-16 | 30 |
| PMT | SMYD3 | BAY-6035 | 2021-06-21 | 27 |
| White_Paper | CACHE | CACHE | 2022-02-15 | 116 |
| USP | USP21 | BAY-805 | 2023-02-20 | 28 |
| UBD | HDAC6 | SGC-UBD253 | 2023-07-21 | 12 |
| Kinase | CDKL5 | SGC-CAF382-1 | 2023-07-25 | 15 |
| Total Citations | 16,622 | |||